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fda_approved_drug_library
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FDA-Approved Drug Library
Product No.: L4200

All compounds in FDA approved drug library have well-characterized biological activity, clear targets, safety, and bioavailability – properties which could dramatically accelerate drug development and optimization. It is an effective and ideal tool for drug repurposing and cell differentiation induction. Detailed information on each compound in this library can help scientists quickly finish drug screening or make quick judgement on cell differentiation mechanism, and create conditions for further investigation on the mechanism of action.

Product No.:L4200
  • A unique collection of 1729 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety confirmed by pre-clinical research evidence and clinical trials;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas: oncology, cardiology, anti-inflammatory, immunology, neuropsychiatry, analgesia etc
  • Structurally diverse, medicinally active, and cell permeable;
  • Rich documentation with structure, target, IC50 value and biological activity description;
  • NMR and HPLC/LCMS validated to ensure high purity.
Compound Service
Our compound library can be flexibly customized!View More
Compound library Consultation
Composition of compound library
Apoptosis (166)
Endogenous Metabolite (130)
Adrenergic Receptor (116)
5-HT Receptor (109)
AChR (81)
Histamine Receptor (75)
HIV Protease (70)
Dopamine Receptor (70)
COX (59)
Sodium Channel (57)
Parasite (56)
Antifungal (54)
DNA/RNA Synthesis (54)
Potassium Channel (48)
Glucocorticoid Receptor (43)
Estrogen/progestogen Receptor (38)
Calcium Channel (36)
Topoisomerase (34)
P450 (34)
Ferroptosis (30)
SARS-CoV (30)
RAAS (27)
Serotonin Transporter (27)
ribosome (27)
VEGFR (25)
c-Kit (25)
Dehydrogenase (24)
Mitophagy (24)
PDE (24)
Microtubule Associated (23)
Nucleoside Antimetabolite/Analog (22)
Antifection (22)
Reverse Transcriptase (22)
HCV Protease (21)
Norepinephrine (21)
Progesterone Receptor (20)
Estrogen Receptor/ERR (20)
PDGFR (20)
HSV (20)
GABA Receptor (20)
Proton pump (17)
PPAR (17)
Reactive Oxygen Species (17)
EGFR (17)
Androgen Receptor (16)
Influenza Virus (16)
ATPase (15)
HBV (15)
Prostaglandin Receptor (15)
FLT (15)
Carbonic Anhydrase (14)
DNA Alkylator/Crosslinker (14)
JAK (14)
MAO (13)
FGFR (13)
Thrombin (13)
Proteasome (12)
Src (12)
Adenosine Receptor (12)
AChE (12)
NF-κB (12)
c-Met/HGFR (11)
Virus Protease (11)
Bcr-Abl (11)
Raf (11)
ROS (11)
Transferase (10)
DHFR (10)
MRP (10)
Tyrosine Kinases (10)
ALK (10)
Monoamine Oxidase (10)
PI3K (9)
Phosphatase (9)
Antifolate (9)
iGluR (9)
Drug Metabolite (9)
SGLT (9)
HDAC (9)
c-RET (9)
HMG-CoA Reductase (9)
NO Synthase (9)
Thyroid hormone receptor(THR) (8)
ABC (8)
PARP (8)
TRP/TRPV Channel (8)
CDK (8)
Opioid Receptor (8)
MMP (8)
GluR (8)
mTOR (8)
P-gp (8)
Retinoid Receptor (8)
P2Y Receptor (7)
Factor Xa (7)
PKC (7)
DNA gyrase (7)
DPP-4 (7)
CaMK (7)
Phospholipase (7)
MEK (7)
DNA Methyltransferase (7)
HIF/HIF Prolyl-Hydroxylase (7)
CAT (6)
LPL Receptor (6)
NMDAR (6)
DNA Alkylation (6)
Endothelin Receptor (6)
Trk receptor (6)
STAT (6)
TAM Receptor (6)
S1P Receptor (6)
Histone Methyltransferase (5)
ERK (5)
Monoamine Transporter (5)
Guanylate cyclase (5)
Hedgehog/Smoothened (5)
IL Receptor (5)
Lipoxygenase (5)
TLR (5)
Nrf2 (5)
GPR (5)
TNF (5)
Neurokinin receptor (5)
Ras (5)
ROS Kinase (5)
CFTR (5)
Integrin (4)
Amino Acids and Derivatives (4)
NADPH (4)
Glutathione Peroxidase (4)
FXR (4)
Annexin A (4)
BTK (4)
Antiviral (4)
AMPK (4)
HIF (4)
AhR (4)
HER (4)
NOS (3)
Reductase (3)
Cell wall (3)
Histone Demethylase (3)
GNRH Receptor (3)
Cysteine Protease (3)
ROCK (3)
Aryl Hydrocarbon Receptor (3)
Gamma-secretase (3)
LDL (3)
MT Receptor (3)
Mitochondrial Metabolism (3)
Molecular Glues (3)
Smo (3)
Isocitrate Dehydrogenase (IDH) (3)
BCL (3)
Fatty Acid Synthase (3)
PAK (3)
IGF-1R (3)
DNA (3)
Akt (3)
GPCR19 (3)
Decarboxylase (3)
Neprilysin (3)
GST (3)
Ligand for E3 Ligase (3)
Hydroxylase (3)
Chloride channel (2)
CRM1 (2)
Ligands for Target Protein for PROTAC (2)
Arginase (2)
Antioxidant (2)
CETP (2)
GSK-3 (2)
Melatonin Receptor (2)
CaSR (2)
Rho (2)
Leukotriene Receptor (2)
Caspase (2)
IRE1 (2)
UGT (2)
P2X Receptor (2)
Na-K-Cl cotransporter (2)
Integrase (2)
CCR (2)
Xanthine Oxidase (2)
Thrombopoietin Receptor (2)
Interleukin (2)
Lipid (2)
Beta-Secretase (2)
PGE Synthase (2)
Glutathione reductase (2)
Free radical scavengers (2)
Ephrin Receptor (2)
GluCls (2)
RSV (2)
Beta Amyloid (2)
c-Fms (2)
Melanocortin Receptor (2)
Adenosine deaminase (2)
CGRP Receptor (2)
Complement System (2)
Gap Junction Protein (2)
Syk (2)
Sigma receptor (2)
Protease-activated Receptor (2)
PKM (2)
NPC1L1 (1)
Hydrogenase (1)
ROR (1)
DNA-PK (1)
p38 MAPK (1)
YAP (1)
RAR/RXR  (1)
JNK (1)
gp120/CD4 (1)
TOPK (1)
VDA (1)
PKA (1)
Wnt/beta-catenin (1)
Serine Protease (1)
CSF-1R (1)
IAP (1)
Myosin (1)
Adiponectin receptor (1)
MTH1 (1)
GRK (1)
Glucagon Receptor (1)
Phosphorylase (1)
GlyT (1)
Glucosidase (1)
Hexokinase (1)
PROTAC Linker (1)
FAAH (1)
Vasopressin Receptor (1)
CXCR (1)
Angiotensin-converting Enzyme (ACE) (1)
Chk (1)
Somatostatin (1)
OX Receptor (1)
ACK (1)
Epigenetic Reader Domain (1)
DUB (1)
Telomerase (1)
TGF-beta/Smad (1)
ATP Citrate Lyase (1)
MAPK (1)
OAT (1)
HSP (1)
STING (1)
Pyroptosis (1)
IκB/IKK (1)
CRISPR/Cas9 (1)
Oxytocin Receptor (1)
Aquaporin (1)
PLK (1)
Platelet aggregation (1)
Anti-infection (1)
NADPH-oxidase (1)
Tyrosinase (1)
NOD-like Receptor (NLR) (1)
Example of compound library information
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE