Drug Metabolite/Impurity Library

Product No.： L5800

Scientists already found that the isomers or metabolites of many existing drugs show biological activity. For example, Levopropoxyphene is an antitussive, approved by FDA, but its enantiomer, Dextropropoxyphene, has an analgesic effect; L-sotalol is alpha-blocker while d-sotalol is antiarrythmic. Currently, knowledge of isomerism has helped us in introducing safer and more effective drug alternatives of the newer as well as existing drugs. These compounds that have rich pharmacological evaluation data are ideal as entry point for drug repurposing.

The TargetMol’s Selected drug metabolites/isomers Library, a unique collection of 197 drug isomers/metabolites with a great diversity, can be used for drug screening.

Product No.：L5800

Product Description

A unique collection of 197 drug isomers/metabolites for high throughput screening (HTS) and high content screening (HCS);
Structurally diverse, medicinally active, and cell permeable;
Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
NMR and HPLC/LCMS validated to ensure high purity and quality;

Compound Service

Our compound library can be flexibly customized！View More

Compound library Consultation

Composition of compound library

Others (128)

Endogenous Metabolite (35)

Apoptosis (9)

Autophagy (8)

DNA/RNA Synthesis (6)

Antibiotic (6)

Amino Acids and Derivatives (5)

Antioxidant (4)

Nucleoside Antimetabolite/Analog (4)

Drug Metabolite (4)

COX (4)

Antibacterial (4)

Estrogen/progestogen Receptor (3)

5-HT Receptor (3)

HIV Protease (2)

Adenosine Receptor (2)

Mitophagy (2)

Factor Xa (2)

Estrogen Receptor/ERR (2)

VEGFR (2)

Adrenergic Receptor (2)

ROS (2)

PDGFR (2)

Aromatase (2)

NF-κB (2)

P450 (2)

AChR (2)

c-Kit (2)

Microtubule Associated (2)

Thyroid hormone receptor(THR) (1)

ATPase (1)

Proton pump (1)

CAT (1)

Dopamine Receptor (1)

p38 MAPK (1)

Dehydrogenase (1)

Antifungal (1)

PI3K (1)

DNA Alkylator/Crosslinker (1)

P2Y Receptor (1)

Histamine Receptor (1)

Glutathione Peroxidase (1)

c-Myc (1)

PPAR (1)

Parasite (1)

Glucokinase (1)

Calcium Channel (1)

Aryl Hydrocarbon Receptor (1)

iGluR (1)

Topoisomerase (1)

PDE (1)

Raf (1)

P2X Receptor (1)

NMDAR (1)

DPP-4 (1)

PAK (1)

IL Receptor (1)

CXCR (1)

Xanthine Oxidase (1)

Lipoxygenase (1)

IGF-1R (1)

Norepinephrine (1)

Androgen Receptor (1)

P-gp (1)

Trk receptor (1)

Nrf2 (1)

GABA Receptor (1)

c-RET (1)

Neurokinin receptor (1)

Sodium Channel (1)

S6 Kinase (1)

Tyrosinase (1)

Imidazoline Receptor (1)

Example of compound library information

Empty	1000025-07-9	1000413-72-8	229005-80-5	1000787-75-6	946387-07-1	1000998-59-3	1175526-27-8	1001288-58-9	1001350-96-4	1001404-83-6	Empty
Empty	Vadadustat	TAK875	TAK-779	Tegobuvir	RN-1734	BMS-687453	AM211	FT011	BMS754807	AAI101	Empty
Empty	1001625-82-6	1001645-58-4	1001753-24-7	1001908-89-9	1002304-34-8	1002-84-2	100291-86-9	100299-08-9	10030-52-1	10040-45-6	Empty
Empty	RPW-24	SRT1720 hydrochloride	INH6	SRT 2183	AMG208	Pentadecanoic acid	Apiopaeonoside	Pemirolast potassium	L-Anserine nitrate salt	Sodium Picosulfate	Empty
Empty	100427-26-7	1004316-88-4	10045-45-1	100462-37-1	1004990-28-6	100-51-6	1005-24-9	1005264-47-0	1005334-57-5	1005342-46-0	Empty
Empty	Lercanidipine	Cobicistat	1-Ethyl-2-benzimidazolinone	ROSIRIDIN	PF-AKT400	Benzyl alcohol	1-Methylnicotinamide chloride	MX69	CVT-10216	LCL161	Empty
Empty	1005491-05-3	100-55-0	1005504-62-0	1005883-72-6	100643-71-8	1007207-67-1	10075-50-0	1007647-73-5	100784-20-1	10083-24-6	Empty
Empty	Tirasemtiv	Roniacol	Rg3039	Z433927330	Desloratadine	CH5132799	5-Bromoindole	Smurf1-IN-A01	Halosulfuron-methyl	Piceatannol	Empty
Empty	100872-83-1	100874-08-6	1009119-64-5	1009119-65-6	100929-71-3	1009298-09-2	1009298-59-2	100929-99-5	1009734-33-1	10097-84-4	Empty
Empty	ML346	SB 4	Daclatasvir	Daclatasvir dihydrochloride	NADPH (tetracyclohexanamine)	AZD8055	Vistusertib	PAβN dihydrochloride	HZ1157	Rotundine	Empty
Empty	1009816-48-1	1009817-63-3	1009820-21-6	100986-85-4	101001-34-7	1010411-21-8	1010-60-2	1011244-68-0	1011301-27-1	1011529-10-4	Empty
Empty	Thiamet G	B-AP15	Silmitasertib	Levofloxacin	Pamicogrel	GSK369796 Dihydrochloride	2-Chloronaphthoquinone	TFAP	Tenovin3	Azvudine	Empty
Empty	101152-94-7	101155-02-6	1011557-82-6	1011-74-1	101-20-2	1012054-59-9	101-21-3	101-26-8	101303-98-4	1013101-36-4	Empty
Empty	Milnacipran hydrochloride	BW-A78U	Tenovin-6	DL-Normetanephrine hydrochloride	Triclocarban	CUDC101	Chlorpropham	Mestinon	Zacopride hydrochloride	PF04691502	Empty
Empty	101-31-5	1013-69-0	1013750-77-0	1013753-99-5	10138-52-0	1013920-15-4	1013937-63-7	1014691-61-2	101477-54-7	101494-95-5	Empty
Empty	L-Hyoscyamine	Noreugenin	ML-030	BC-1382	Gadolinium chloride	Vorolanib	VTP-27999 TFA	GSK0660	Lomerizine hydrochloride	8-CHLOROQUINAZOLIN-4(1H)-ONE	Empty

Specification	Special Discount Waiting for you to inquire！
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