Clinical Compound Library

Product No.： L3400

Clinical compound library is a collection of 3404 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

Product No.：L3400

Product Description

A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
An effective tool for new drug screening and cell differentiation induction;
Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
Structurally diverse, medicinally active, and cell permeable;
NMR and HPLC validated to ensure high purity and quality;

Compound Service

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Compound library Consultation

Composition of compound library

5-HT Receptor (145)

Adrenergic Receptor (109)

DNA/RNA Synthesis (98)

HIV Protease (92)

AChR (90)

Dopamine Receptor (88)

COX (84)

VEGFR (77)

Histamine Receptor (76)

Parasite (71)

Sodium Channel (66)

Calcium Channel (64)

EGFR (64)

PI3K (63)

Antifungal (62)

Potassium Channel (60)

PDE (59)

FLT (56)

Topoisomerase (55)

CDK (52)

HCV Protease (51)

PDGFR (50)

P450 (50)

JAK (46)

c-Kit (46)

Dehydrogenase (44)

PPAR (44)

Reactive Oxygen Species (44)

FGFR (44)

Microtubule Associated (44)

SARS-CoV (43)

Ferroptosis (42)

HDAC (42)

Glucocorticoid Receptor (41)

mTOR (41)

c-Met/HGFR (39)

Influenza Virus (39)

Estrogen/progestogen Receptor (35)

Src (34)

Mitophagy (34)

NF-κB (34)

RAAS (33)

Prostaglandin Receptor (33)

GABA Receptor (33)

HBV (32)

Nucleoside Antimetabolite/Analog (31)

Reverse Transcriptase (31)

Tyrosine Kinases (29)

GPR (28)

Adenosine Receptor (27)

Bcr-Abl (26)

Proteasome (25)

Raf (25)

BTK (25)

Androgen Receptor (25)

PARP (23)

Serotonin Transporter (23)

iGluR (23)

Akt (23)

HER (23)

Aurora Kinase (22)

Epigenetic Reader Domain (22)

Virus Protease (21)

ROS (21)

Opioid Receptor (21)

HSV (21)

MEK (21)

Transferase (20)

Norepinephrine (20)

Phosphatase (19)

Progesterone Receptor (19)

Estrogen Receptor/ERR (19)

IL Receptor (19)

GluR (19)

HSP (19)

p38 MAPK (18)

ALK (18)

Beta Amyloid (18)

c-RET (18)

TNF (18)

HIF/HIF Prolyl-Hydroxylase (18)

ERK (17)

Antifection (17)

DPP-4 (17)

P-gp (17)

Trk receptor (17)

ATPase (16)

Carbonic Anhydrase (16)

Antioxidant (16)

DNA Alkylator/Crosslinker (16)

TRP/TRPV Channel (16)

NMDAR (16)

ribosome (16)

GSK-3 (15)

PKC (15)

AChE (15)

c-Fms (15)

Thrombin (15)

Proton pump (14)

Gamma-secretase (14)

Mitochondrial Metabolism (14)

CXCR (14)

Endothelin Receptor (14)

Interleukin (14)

TLR (14)

Retinoid Receptor (14)

TAM Receptor (14)

DNA-PK (13)

MAO (13)

E1/E2/E3 Enzyme (13)

BCL (13)

CCR (13)

MMP (13)

Chk (13)

Antiviral (13)

STAT (13)

AMPK (13)

Phospholipase (13)

Histone Methyltransferase (12)

LPL Receptor (12)

Caspase (12)

SGLT (12)

HIF (12)

Syk (12)

NO Synthase (12)

S1P Receptor (12)

Thyroid hormone receptor(THR) (11)

Antifolate (11)

Guanylate cyclase (11)

DNA Alkylation (11)

CFTR (11)

p53 (11)

Integrin (10)

NADPH (10)

CSF-1R (10)

Hedgehog/Smoothened (10)

IGF-1R (10)

Nrf2 (10)

CETP (9)

Glutathione Peroxidase (9)

MRP (9)

PKA (9)

Wnt/beta-catenin (9)

P2X Receptor (9)

Lipoxygenase (9)

TGF-beta/Smad (9)

Hydroxylase (9)

PLK (9)

Cannabinoid Receptor (9)

HMG-CoA Reductase (9)

S6 Kinase (9)

FAK (9)

Monoamine Oxidase (9)

DHFR (8)

P2Y Receptor (8)

Reductase (8)

JNK (8)

GNRH Receptor (8)

ROCK (8)

IAP (8)

Drug Metabolite (8)

Glucosidase (8)

Vasopressin Receptor (8)

OX Receptor (8)

Indoleamine 2,3-Dioxygenase (IDO) (8)

Sirtuin (8)

Casein Kinase (8)

ATM/ATR (8)

Neurokinin receptor (8)

Ras (8)

ROS Kinase (8)

Mdm2 (7)

CAT (7)

Histone Demethylase (7)

Pim (7)

Serine Protease (7)

FXR (7)

Aryl Hydrocarbon Receptor (7)

Smo (7)

Xanthine Oxidase (7)

Beta-Secretase (7)

Aminopeptidase (7)

RSV (7)

DNA Methyltransferase (7)

Sigma receptor (7)

Kinesin (7)

ROR (6)

Amino Acids and Derivatives (6)

BACE (6)

Glucokinase (6)

RIP kinase (6)

Isocitrate Dehydrogenase (IDH) (6)

PAK (6)

Bradykinin Receptor (6)

DNA (6)

IκB/IKK (6)

Ligand for E3 Ligase (6)

IRAK (6)

AhR (6)

Tie-2 (5)

Factor Xa (5)

Leukotriene Receptor (5)

IDO (5)

Glucagon Receptor (5)

DNA gyrase (5)

Fatty Acid Synthase (5)

Acyltransferase (5)

Ephrin Receptor (5)

Complement System (5)

Chloride channel (4)

NOS (4)

DprE1 (4)

LTR (4)

IFNAR (4)

Melatonin Receptor (4)

Liver X Receptor (4)

MT Receptor (4)

Monoamine Transporter (4)

Molecular Glues (4)

FAAH (4)

KSP (4)

CaMK (4)

Wee1 (4)

PGE Synthase (4)

Decarboxylase (4)

CRFR (4)

Neprilysin (4)

Acetyl-CoA Carboxylase (4)

GHSR (4)

CGRP Receptor (4)

Gap Junction Protein (4)

NADPH-oxidase (4)

cholecystokinin (4)

CRM1 (3)

Arginase (3)

YAP (3)

Cell wall (3)

ABC (3)

CaSR (3)

Rho (3)

Serine/threonin kinase (3)

Cysteine Protease (3)

NAMPT (3)

Myosin (3)

Annexin A (3)

GlyT (3)

Neuropeptide Y Receptor (3)

Somatostatin (3)

DUB (3)

Telomerase (3)

OAT (3)

STING (3)

Free radical scavengers (3)

GPCR19 (3)

LPA Receptor (3)

Melanocortin Receptor (3)

PDK (3)

Adenosine deaminase (3)

Tyrosinase (3)

Protease-activated Receptor (3)

NOD-like Receptor (NLR) (3)

Imidazoline Receptor (3)

PD-1/PD-L1 (3)

Taste receptor (2)

NEDD8 (2)

Ligands for Target Protein for PROTAC (2)

PERK (2)

VDA (2)

Galectin (2)

PYK2 (2)

IRE1 (2)

UGT (2)

LDL (2)

Na-K-Cl cotransporter (2)

Hexokinase (2)

Integrase (2)

Stearoyl-CoA Desaturase (SCD) (2)

Epoxide Hydrolase (2)

ATP Citrate Lyase (2)

Lipid (2)

BCRP (2)

MAPK (2)

Porcupine (2)

CD73 (2)

transporter (2)

PAI-1 (2)

GST (2)

Oxytocin Receptor (2)

Discoidin Domain Receptor (DDR) (2)

p97 (2)

MLK (2)

advanced glycation end products (1)

Adenylyl cyclase (1)

PROTACs (1)

GSNOR (1)

NPC1L1 (1)

Monocarboxylate transporter (1)

Hydrogenase (1)

MALT (1)

Arrestin (1)

RAR/RXR (1)

DYRK (1)

Lipase (1)

TOPK (1)

GTPase (1)

c-Myc (1)

N-Acetylglucosaminyltransferase (1)

VDAC (1)

Hck (1)

Stemness kinase (1)

Glutaminase (1)

FLAP (1)

Motilin Receptor (1)

PAFR (1)

MTH1 (1)

Fas/FasL (1)

GRK (1)

Phosphorylase (1)

AAK1 (AP2 associated kinase 1) (1)

Anion Exchanger (1)

PROTAC Linker (1)

HCN Channel (1)

Thioredoxin (1)

ACK (1)

MNK (1)

Survivin (1)

Histone Acetyltransferase (1)

ASK (1)

GluCls (1)

Pyroptosis (1)

MELK (1)

Methionine Adenosyltransferase (MAT) (1)

Hippo pathway (1)

Aromatase (1)

KLF (1)

PI4K (1)

CRISPR/Cas9 (1)

Aquaporin (1)

SGK (1)

Anti-infection (1)

NOD (1)

BMI-1 (1)

PKM (1)

Example of compound library information

Empty	1000025-07-9	1000413-72-8	229005-80-5	1000787-75-6	946387-07-1	1000998-59-3	1175526-27-8	1001288-58-9	1001350-96-4	1001404-83-6	Empty
Empty	Vadadustat	TAK875	TAK-779	Tegobuvir	RN-1734	BMS-687453	AM211	FT011	BMS754807	AAI101	Empty
Empty	1001625-82-6	1001645-58-4	1001753-24-7	1001908-89-9	1002304-34-8	1002-84-2	100291-86-9	100299-08-9	10030-52-1	10040-45-6	Empty
Empty	RPW-24	SRT1720 hydrochloride	INH6	SRT 2183	AMG208	Pentadecanoic acid	Apiopaeonoside	Pemirolast potassium	L-Anserine nitrate salt	Sodium Picosulfate	Empty
Empty	100427-26-7	1004316-88-4	10045-45-1	100462-37-1	1004990-28-6	100-51-6	1005-24-9	1005264-47-0	1005334-57-5	1005342-46-0	Empty
Empty	Lercanidipine	Cobicistat	1-Ethyl-2-benzimidazolinone	ROSIRIDIN	PF-AKT400	Benzyl alcohol	1-Methylnicotinamide chloride	MX69	CVT-10216	LCL161	Empty
Empty	1005491-05-3	100-55-0	1005504-62-0	1005883-72-6	100643-71-8	1007207-67-1	10075-50-0	1007647-73-5	100784-20-1	10083-24-6	Empty
Empty	Tirasemtiv	Roniacol	Rg3039	Z433927330	Desloratadine	CH5132799	5-Bromoindole	Smurf1-IN-A01	Halosulfuron-methyl	Piceatannol	Empty
Empty	100872-83-1	100874-08-6	1009119-64-5	1009119-65-6	100929-71-3	1009298-09-2	1009298-59-2	100929-99-5	1009734-33-1	10097-84-4	Empty
Empty	ML346	SB 4	Daclatasvir	Daclatasvir dihydrochloride	NADPH (tetracyclohexanamine)	AZD8055	Vistusertib	PAβN dihydrochloride	HZ1157	Rotundine	Empty
Empty	1009816-48-1	1009817-63-3	1009820-21-6	100986-85-4	101001-34-7	1010411-21-8	1010-60-2	1011244-68-0	1011301-27-1	1011529-10-4	Empty
Empty	Thiamet G	B-AP15	Silmitasertib	Levofloxacin	Pamicogrel	GSK369796 Dihydrochloride	2-Chloronaphthoquinone	TFAP	Tenovin3	Azvudine	Empty
Empty	101152-94-7	101155-02-6	1011557-82-6	1011-74-1	101-20-2	1012054-59-9	101-21-3	101-26-8	101303-98-4	1013101-36-4	Empty
Empty	Milnacipran hydrochloride	BW-A78U	Tenovin-6	DL-Normetanephrine hydrochloride	Triclocarban	CUDC101	Chlorpropham	Mestinon	Zacopride hydrochloride	PF04691502	Empty
Empty	101-31-5	1013-69-0	1013750-77-0	1013753-99-5	10138-52-0	1013920-15-4	1013937-63-7	1014691-61-2	101477-54-7	101494-95-5	Empty
Empty	L-Hyoscyamine	Noreugenin	ML-030	BC-1382	Gadolinium chloride	Vorolanib	VTP-27999 TFA	GSK0660	Lomerizine hydrochloride	8-CHLOROQUINAZOLIN-4(1H)-ONE	Empty

Specification	Special Discount Waiting for you to inquire！
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