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bioactive_lipid_compound_library
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Bioactive Lipid Compound Library
Product No.: L7000

Bioactive lipids have been shown to provide health benefits either through modification of tissue fatty acid composition or induction of cell signaling pathways, due to their pivotal role in immune regulation, inflammation, and maintenance of tissue homeostasis. While some health benefits are derived from consumption of short to medium-chain fatty acids, evidence suggests that the polyunsaturated fatty acids (PUFAs) are the most important bioactive lipids. PUFAs are found mostly in plant seed oils and are important substrates for the biosynthesis of cellular hormones (eicosanoids) and other signaling compounds that modulate human health. The beneficial health effects of PUFAs seem to be dependent on their isomer configuration as the cis-isomer is the predominant bioactive form which enhances membrane fluidity when incorporated into cells. Increased membrane fluidity enhances cell to cell communication and helps maintain normal homeostasis or prevent the development of metabolic disorders.

The TargetMol’s Bioactive Lipid Inhibitor Library, a unique collection of 385 bioactive lipids related compounds, can be used for research in bioactive lipids, and high throughput screening (HTS) and high content screening (HCS).

Product No.:L7000
  • A unique collection of 385 bioactive lipids related compounds for high throughput screening (HTS) and high content screening (HCS), including Agonists & Antagonists, Endocannabinoids, Farnesyl/geranylgeranyl derivates, HETEs deHETEs, hepoxilins, Polyunsaturated fatty acids, Leukotrienes, lipoxins, LPA & phosphatidic acids, Octadecanoids, PAFs, Prostaglandins & thromboxanes, Retinoids, vitamin D metabolites, Sphingolipids, etc.;
  • Targets include GPCR, HDAC, PPAR, DNA Alkylating, EGFR, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;
Compound Service
Our compound library can be flexibly customized!View More
Compound library Consultation
Composition of compound library
Endogenous Metabolite (91)
Autophagy (82)
Others (59)
Apoptosis (53)
PDE (48)
COX (25)
PPAR (20)
Estrogen/progestogen Receptor (19)
Antibacterial (18)
Phospholipase (17)
MAO (15)
Ferroptosis (13)
TRP/TRPV Channel (11)
Antifungal (10)
Lipoxygenase (10)
Prostaglandin Receptor (10)
P450 (10)
HMG-CoA Reductase (10)
HIV Protease (9)
Mitophagy (9)
HDAC (9)
Thrombin (9)
Adenosine Receptor (8)
Estrogen Receptor/ERR (8)
FXR (8)
Glucocorticoid Receptor (8)
NF-κB (8)
Cannabinoid Receptor (8)
Antibiotic (8)
Monoamine Oxidase (8)
PI3K (7)
Lipase (7)
Reactive Oxygen Species (7)
Retinoid Receptor (7)
Potassium Channel (7)
Factor Xa (6)
Virus Protease (6)
Fatty Acid Synthase (6)
Lipid (6)
TNF (6)
AhR (6)
Dehydrogenase (5)
Progesterone Receptor (5)
Parasite (5)
Calcium Channel (5)
Adrenergic Receptor (5)
Aryl Hydrocarbon Receptor (5)
Sirtuin (5)
Casein Kinase (5)
AChR (5)
p38 MAPK (4)
CETP (4)
Histamine Receptor (4)
PKC (4)
Nrf2 (4)
Influenza Virus (4)
GPR (4)
GABA Receptor (4)
Antioxidant (3)
Phosphatase (3)
Liver X Receptor (3)
FAAH (3)
Androgen Receptor (3)
Akt (3)
DNA/RNA Synthesis (3)
GPCR19 (3)
IκB/IKK (3)
5-HT Receptor (3)
PLK (3)
HIF (3)
Sodium Channel (3)
p53 (3)
Mdm2 (2)
Chloride channel (2)
DNA-PK (2)
LPL Receptor (2)
LTR (2)
Histone Demethylase (2)
Glutathione Peroxidase (2)
GSK-3 (2)
MRP (2)
PARP (2)
Leukotriene Receptor (2)
Caspase (2)
ERK (2)
LDL (2)
CDK (2)
Mitochondrial Metabolism (2)
ROS (2)
Opioid Receptor (2)
BCL (2)
PAK (2)
MMP (2)
CaMK (2)
DNA (2)
mTOR (2)
TGF-beta/Smad (2)
AChE (2)
Acyltransferase (2)
RSV (2)
LPA Receptor (2)
Proteasome (1)
ATPase (1)
NOS (1)
Transferase (1)
Monocarboxylate transporter (1)
Dopamine Receptor (1)
ROR (1)
Src (1)
c-Met/HGFR (1)
DNA Alkylator/Crosslinker (1)
Reductase (1)
DYRK (1)
NADPH (1)
Melatonin Receptor (1)
ABC (1)
PKA (1)
HBV (1)
Tyrosine Kinases (1)
Wnt/beta-catenin (1)
Nucleoside Antimetabolite/Analog (1)
Cysteine Protease (1)
VEGFR (1)
iGluR (1)
IAP (1)
Topoisomerase (1)
Annexin A (1)
RIP kinase (1)
UGT (1)
Gamma-secretase (1)
Drug Metabolite (1)
Phosphorylase (1)
P2X Receptor (1)
NMDAR (1)
Guanylate cyclase (1)
Smo (1)
PDGFR (1)
Hedgehog/Smoothened (1)
HSV (1)
IL Receptor (1)
PAD (1)
Xanthine Oxidase (1)
Epoxide Hydrolase (1)
GluR (1)
Epigenetic Reader Domain (1)
EGFR (1)
PGE Synthase (1)
MNK (1)
P-gp (1)
HSP (1)
SARS-CoV (1)
Histone Acetyltransferase (1)
PAI-1 (1)
ALK (1)
ATM/ATR (1)
Acetyl-CoA Carboxylase (1)
STAT (1)
AMPK (1)
Hydroxylase (1)
MEK (1)
c-RET (1)
Platelet aggregation (1)
NADPH-oxidase (1)
NOD (1)
Ras (1)
Tyrosinase (1)
Microtubule Associated (1)
FAK (1)
HIF/HIF Prolyl-Hydroxylase (1)
MLK (1)
PKM (1)
S1P Receptor (1)
NO Synthase (1)
Example of compound library information
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE