Anti-Cancer Drug Library

Product No.： L2150

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 3080 anticancer drugs including FDA approved and compounds in clinical trial phases as Anticancer Drug Library that can be used for tumor-related research and anti-tumor drug screening.

Product No.：L2150

Product Description

A unique collection of 3080 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
Structurally diverse, medicinally active, and cell permeable;
NMR and HPLC validated to ensure high purity and quality;

Compound Service

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Compound library Consultation

Composition of compound library

Endogenous Metabolite (173)

Adrenergic Receptor (169)

Antibacterial (144)

COX (135)

Dopamine Receptor (126)

Histamine Receptor (125)

Antibiotic (119)

DNA/RNA Synthesis (116)

Sodium Channel (95)

Calcium Channel (86)

Potassium Channel (85)

VEGFR (81)

EGFR (76)

AChR (72)

Parasite (68)

PI3K (65)

Glucocorticoid Receptor (61)

Reactive Oxygen Species (61)

P450 (58)

FLT (55)

HIV Protease (53)

Topoisomerase (53)

CDK (53)

NF-κB (53)

PDGFR (52)

PPAR (51)

GABA Receptor (49)

JAK (48)

c-Kit (48)

FGFR (46)

HDAC (44)

Ferroptosis (42)

Prostaglandin Receptor (42)

Estrogen/progestogen Receptor (41)

Antifungal (41)

mTOR (41)

Microtubule Associated (41)

c-Met/HGFR (40)

Dehydrogenase (39)

Mitophagy (38)

Influenza Virus (37)

Estrogen Receptor/ERR (36)

Src (34)

Nucleoside Antimetabolite/Analog (34)

iGluR (32)

SARS-CoV (32)

Adenosine Receptor (31)

Tyrosine Kinases (31)

Androgen Receptor (31)

PDE (30)

GPR (30)

Opioid Receptor (29)

Bcr-Abl (28)

Raf (28)

Serotonin Transporter (25)

HER (25)

ATPase (24)

Norepinephrine (24)

Akt (24)

PARP (23)

Aurora Kinase (23)

TRP/TRPV Channel (22)

p38 MAPK (21)

HSV (21)

Epigenetic Reader Domain (21)

P-gp (21)

MEK (21)

TNF (21)

Proton pump (20)

Virus Protease (20)

PKC (20)

NMDAR (20)

BTK (20)

HSP (20)

DNA Alkylator/Crosslinker (19)

RAAS (18)

ERK (18)

ALK (18)

HIF/HIF Prolyl-Hydroxylase (18)

HBV (17)

ROS (17)

Trk receptor (17)

c-RET (17)

HCV Protease (16)

Phosphatase (16)

GSK-3 (16)

CXCR (16)

AMPK (16)

Carbonic Anhydrase (15)

GNRH Receptor (15)

Caspase (15)

Drug Metabolite (15)

BCL (15)

Endothelin Receptor (15)

MMP (15)

SGLT (15)

Histone Methyltransferase (14)

Progesterone Receptor (14)

Retinoid Receptor (14)

STAT (14)

c-Fms (14)

TAM Receptor (14)

Proteasome (13)

DNA-PK (13)

E1/E2/E3 Enzyme (13)

Guanylate cyclase (13)

IL Receptor (13)

Chk (13)

Reverse Transcriptase (13)

LPL Receptor (12)

MAO (12)

DNA Alkylation (12)

TGF-beta/Smad (12)

HIF (12)

CFTR (12)

p53 (12)

S1P Receptor (12)

Transferase (11)

DHFR (11)

MRP (11)

PKA (11)

Antifolate (11)

Gamma-secretase (11)

P2X Receptor (11)

Mitochondrial Metabolism (11)

Hedgehog/Smoothened (11)

GluR (11)

Lipoxygenase (11)

IGF-1R (11)

Interleukin (11)

Cannabinoid Receptor (11)

Neurokinin receptor (11)

HMG-CoA Reductase (11)

Monoamine Oxidase (11)

Antioxidant (10)

P2Y Receptor (10)

Wnt/beta-catenin (10)

ROCK (10)

Vasopressin Receptor (10)

AChE (10)

Nrf2 (10)

Syk (10)

FAK (10)

Chloride channel (9)

IAP (9)

CSF-1R (9)

Antifection (9)

Indoleamine 2,3-Dioxygenase (IDO) (9)

TLR (9)

Beta Amyloid (9)

S6 Kinase (9)

NADPH (8)

JNK (8)

Smo (8)

OX Receptor (8)

CaMK (8)

Casein Kinase (8)

ATM/ATR (8)

Phospholipase (8)

PLK (8)

DNA Methyltransferase (8)

Ras (8)

Sigma receptor (8)

ROS Kinase (8)

Mdm2 (7)

Integrin (7)

ABC (7)

Pim (7)

Glucagon Receptor (7)

Monoamine Transporter (7)

Antiviral (7)

Sirtuin (7)

Ligand for E3 Ligase (7)

Aromatase (7)

cholecystokinin (7)

Thrombin (7)

Kinesin (7)

Histone Demethylase (6)

Glutathione Peroxidase (6)

Leukotriene Receptor (6)

RIP kinase (6)

Isocitrate Dehydrogenase (IDH) (6)

PAK (6)

CCR (6)

Bradykinin Receptor (6)

DNA (6)

IκB/IKK (6)

IRAK (6)

NO Synthase (6)

IFNAR (5)

Tie-2 (5)

Serine Protease (5)

FXR (5)

DPP-4 (5)

Fatty Acid Synthase (5)

PGE Synthase (5)

GPCR19 (5)

Ephrin Receptor (5)

ribosome (5)

GHSR (5)

Hydroxylase (5)

NOD (5)

Amino Acids and Derivatives (4)

LTR (4)

Melatonin Receptor (4)

CaSR (4)

Serine/threonin kinase (4)

Aryl Hydrocarbon Receptor (4)

IDO (4)

Annexin A (4)

Molecular Glues (4)

Somatostatin (4)

Xanthine Oxidase (4)

KSP (4)

Wee1 (4)

Aminopeptidase (4)

CRFR (4)

Melanocortin Receptor (4)

PDK (4)

Oxytocin Receptor (4)

CGRP Receptor (4)

Tyrosinase (4)

AhR (4)

PD-1/PD-L1 (4)

Monocarboxylate transporter (3)

ROR (3)

CRM1 (3)

YAP (3)

Reductase (3)

Rho (3)

Cysteine Protease (3)

Liver X Receptor (3)

NAMPT (3)

UGT (3)

MT Receptor (3)

DNA gyrase (3)

Na-K-Cl cotransporter (3)

Hexokinase (3)

Neuropeptide Y Receptor (3)

DUB (3)

MAPK (3)

OAT (3)

STING (3)

Free radical scavengers (3)

RSV (3)

GST (3)

Adenosine deaminase (3)

Protease-activated Receptor (3)

NOD-like Receptor (NLR) (3)

PROTACs (2)

NOS (2)

CAT (2)

NEDD8 (2)

Ligands for Target Protein for PROTAC (2)

Arginase (2)

Cell wall (2)

PERK (2)

Factor Xa (2)

VDA (2)

PYK2 (2)

IRE1 (2)

LDL (2)

Glucosidase (2)

PROTAC Linker (2)

Telomerase (2)

Lipid (2)

ATP Citrate Lyase (2)

BCRP (2)

Beta-Secretase (2)

Acyltransferase (2)

Porcupine (2)

CD73 (2)

transporter (2)

Decarboxylase (2)

LPA Receptor (2)

Gap Junction Protein (2)

Discoidin Domain Receptor (DDR) (2)

p97 (2)

MLK (2)

Imidazoline Receptor (2)

advanced glycation end products (1)

NPC1L1 (1)

Hydrogenase (1)

MALT (1)

Na+/Ca2+ Exchanger (1)

BACE (1)

DYRK (1)

RAR/RXR (1)

Lipase (1)

TOPK (1)

GTPase (1)

Galectin (1)

c-Myc (1)

Kisspeptin (1)

N-Acetylglucosaminyltransferase (1)

Hck (1)

Glucokinase (1)

Stemness kinase (1)

Glutaminase (1)

Immunology/Inflammation related (1)

Myosin (1)

Motilin Receptor (1)

Adiponectin receptor (1)

PAFR (1)

MTH1 (1)

GRK (1)

GlyT (1)

Anion Exchanger (1)

HCN Channel (1)

Thioredoxin (1)

FAAH (1)

PAD (1)

ACK (1)

cAMP (1)

Thrombopoietin Receptor (1)

Glutathione reductase (1)

Survivin (1)

MNK (1)

Histone Acetyltransferase (1)

ASK (1)

GluCls (1)

PAI-1 (1)

Pyroptosis (1)

MELK (1)

Methionine Adenosyltransferase (MAT) (1)

Hippo pathway (1)

Neprilysin (1)

PI4K (1)

KLF (1)

Aquaporin (1)

SGK (1)

Complement System (1)

Platelet aggregation (1)

NADPH-oxidase (1)

BMI-1 (1)

Example of compound library information

Empty	1000025-07-9	1000413-72-8	229005-80-5	1000787-75-6	946387-07-1	1000998-59-3	1175526-27-8	1001288-58-9	1001350-96-4	1001404-83-6	Empty
Empty	Vadadustat	TAK875	TAK-779	Tegobuvir	RN-1734	BMS-687453	AM211	FT011	BMS754807	AAI101	Empty
Empty	1001625-82-6	1001645-58-4	1001753-24-7	1001908-89-9	1002304-34-8	1002-84-2	100291-86-9	100299-08-9	10030-52-1	10040-45-6	Empty
Empty	RPW-24	SRT1720 hydrochloride	INH6	SRT 2183	AMG208	Pentadecanoic acid	Apiopaeonoside	Pemirolast potassium	L-Anserine nitrate salt	Sodium Picosulfate	Empty
Empty	100427-26-7	1004316-88-4	10045-45-1	100462-37-1	1004990-28-6	100-51-6	1005-24-9	1005264-47-0	1005334-57-5	1005342-46-0	Empty
Empty	Lercanidipine	Cobicistat	1-Ethyl-2-benzimidazolinone	ROSIRIDIN	PF-AKT400	Benzyl alcohol	1-Methylnicotinamide chloride	MX69	CVT-10216	LCL161	Empty
Empty	1005491-05-3	100-55-0	1005504-62-0	1005883-72-6	100643-71-8	1007207-67-1	10075-50-0	1007647-73-5	100784-20-1	10083-24-6	Empty
Empty	Tirasemtiv	Roniacol	Rg3039	Z433927330	Desloratadine	CH5132799	5-Bromoindole	Smurf1-IN-A01	Halosulfuron-methyl	Piceatannol	Empty
Empty	100872-83-1	100874-08-6	1009119-64-5	1009119-65-6	100929-71-3	1009298-09-2	1009298-59-2	100929-99-5	1009734-33-1	10097-84-4	Empty
Empty	ML346	SB 4	Daclatasvir	Daclatasvir dihydrochloride	NADPH (tetracyclohexanamine)	AZD8055	Vistusertib	PAβN dihydrochloride	HZ1157	Rotundine	Empty
Empty	1009816-48-1	1009817-63-3	1009820-21-6	100986-85-4	101001-34-7	1010411-21-8	1010-60-2	1011244-68-0	1011301-27-1	1011529-10-4	Empty
Empty	Thiamet G	B-AP15	Silmitasertib	Levofloxacin	Pamicogrel	GSK369796 Dihydrochloride	2-Chloronaphthoquinone	TFAP	Tenovin3	Azvudine	Empty
Empty	101152-94-7	101155-02-6	1011557-82-6	1011-74-1	101-20-2	1012054-59-9	101-21-3	101-26-8	101303-98-4	1013101-36-4	Empty
Empty	Milnacipran hydrochloride	BW-A78U	Tenovin-6	DL-Normetanephrine hydrochloride	Triclocarban	CUDC101	Chlorpropham	Mestinon	Zacopride hydrochloride	PF04691502	Empty
Empty	101-31-5	1013-69-0	1013750-77-0	1013753-99-5	10138-52-0	1013920-15-4	1013937-63-7	1014691-61-2	101477-54-7	101494-95-5	Empty
Empty	L-Hyoscyamine	Noreugenin	ML-030	BC-1382	Gadolinium chloride	Vorolanib	VTP-27999 TFA	GSK0660	Lomerizine hydrochloride	8-CHLOROQUINAZOLIN-4(1H)-ONE	Empty

Specification	Special Discount Waiting for you to inquire！
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